BIBU 1361 dihydrochloride

BIBU 1361 dihydrochloride (订货以CAS编码或英文名称为准)

EGFR抑制剂BIBU1361 is a potent, selective, orally active EGFR inhibitor with IC50 of 3 nM, shows weak activity against HER2 (IC50=280 nM) and no inhibition on IGF1R, HGFR, Src, and VEGFR2 (IC50>10 uM).
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编号:MED19444
分子式:C22H27N7FCL.2[HCL]
CAS号:793726-84-8
分子量:516.87
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MED19444-1mg MedBio 1mg ≥98% ¥3765.00 登录后可见
英文名称: BIBU 1361 dihydrochloride
CAS号: 793726-84-8
分子式: C22H27N7FCL.2[HCL]
分子量: 516.87
EGFR抑制剂BIBU1361 is a potent, selective, orally active EGFR inhibitor with IC50 of 3 nM, shows weak activity against HER2 (IC50=280 nM) and no inhibition on IGF1R, HGFR, Src, and VEGFR2 (IC50>10 uM).
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