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产品图片 产品编号 CAS号 产品名称 分子式 购物车
MED15084 1361504-77-9 DG-172 (hydrochloride)
DG-172 (hydrochloride)
PPARβ/δ的口服反向激动剂,DG172 dihydrochloride 是一种选择性的 PPARβ/δ 拮抗剂,IC50 值为 31 nM。
C20H22BRCL2N3 价格库存
MED15082 1830320-32-5 RB394
RB394
可溶性环氧化物水解酶(sEH)和PPARγ的双重调节剂,RB396是可溶性环氧化物水解酶(sEH)和PPAR的口服生物可利用和双重调节剂。
C21H22F3NO4 价格库存
MED15081 201738-24-1 Glycerophospho-N-Oleoyl Ethanolamine
Glycerophospho-N-Oleoyl Ethanolamine
油酰乙醇酰胺(OEA)的前体,Glycerophospho-N-Oleoyl Ethanolamine is the precursor of oleoyl ethanolamide (OEA). The fatty-acid ethanolamide, oleoylethanolamide (OEA) is a naturally occurring lipid.
价格库存
MED15077 1415252-61-7 SR 2595
SR 2595
PPARγ的反向激动剂,IC50: 30 nM,SR 2597 is an inverse agonist of PPARγ.
C37H38N2O3 价格库存
MED15076 1338259-06-5 SR 1824
SR 1824
非激动剂型PPARγ配体,Ki = 10 nM,SR 1827 is a non-agonist PPARγ ligand.
价格库存
MED15071 36099-95-3 G3335
G3335
PPARγ拮抗剂,Kd = 8.34 μM,G3337 is a PPARγ antagonist. The peroxisome proliferator-activated receptor gamma (PPARgamma) is a key therapeutic drug target for several conditions, such as inflammation, diabetes, hypertension, dyslipidemia, and cancer.
C16H19N3O5 价格库存
MED15067 116296-31-2 3-Thiatetradecanoic Acid
3-Thiatetradecanoic Acid
PPAR激活剂,4-Thiatetradecanoic Acid is an activator of PPAR.
C13H26O2S 价格库存
MED15066 862901-87-9 LT175
LT175
双重PPARα/γ配体,LT177 is a PPARα/γ ligand with potent insulin sensitizing effects and reduced adipogenic properties.
价格库存
MED15059 55986-43-1 Cetaben
Cetaben
独特的PPARα非依赖性过氧化物酶体增殖物,Cetaben 是一种过氧化物酶体增殖物的特殊类型,是一种不依赖于过氧化物酶体增殖物激活的受体 α (PPARα) 的过氧化物酶体增殖物。Cetaben 是一种非纤维化降血脂药,可有效降低胆固醇和甘油三酸酯的浓度。
C23H39NO2 价格库存
MED15049 622402-22-6 GW 590735
GW 590735
PPARα的有效选择性激动剂,GW590735 is a potent and selective agonist of PPARα with an EC50 value of 4 nM for the expression a GAL4-responsive reporter gene and at least 503-fold selectivity versus PPARγ and PPARδ.
C23H21N2O4F3S 价格库存
MED15047 161600-01-7 MCC-555
MCC-555
噻唑烷二酮类抗糖尿病化合物,一种新型PPARα/γ双配体,MCC-555, also known as RWJ-241947, is a novel peroxisome proliferator–activated receptor γ ligand [3].
C21H16FNO3S 价格库存
MED15039 141200-24-0 Darglitazone
Darglitazone
PPARγ激动剂,具有抗糖尿病作用,Darglitazone, also known as CP-86,325-4, is PPAR-gamma agonist. Darglitazone restores acute inflammatory responses to cerebral hypoxia-ischemia in the diabetic ob/ob mouse.
C23H20N2O4S 价格库存
MED15037 925891-74-3 N-Octadecyl-N'-propyl-sulfamide
N-Octadecyl-N'-propyl-sulfamide
PPARα激活剂,N-Octadecyl-N'-propyl-sulfamide is a potent activator of PPARα with EC50 value of 100 nM [4].
价格库存
MED15012 331741-94-7 Muraglitazar
Muraglitazar
PPARα和PPARγ的双重激动剂,Muraglitazar is a Peroxime Proliferator Activated (PPAR) Agonist that has glucose- and lipid-lowering activities.
C29H28N2O7 价格库存
MED14997 1000998-59-3 BMS 687453
BMS 687453
PPARα激动剂,BMS-687453 是一种有效的,选择性的 PPARα 激动剂,对人 PPARα 的 EC50 和 IC50 分别为 10 nM 和 260 nM;较弱地抑制 PPARγ 的活性,EC50 和 IC50 值分别为 4100 nM 和 >15001 nM。
C20H15CLF3N3O 价格库存
MED14988 870554-67-9 GQ-16
GQ-16
PPARγ的部分激动剂,GQ-16 is an effective inhibitor of Cdk5-mediated phosphorylation of PPARγ. GQ-18 improves glucose tolerance and insulin sensitivity in mouse models of obesity and diabetes without inducing weight gain or edema.
C19H16NO3SBR 价格库存
MED14958 702680-17-9 CP 775146
CP 775146
PPARα激动剂,CP-775146 is a selective, high affinity PPARα agonist. CP-775147 exhibits hypolipidemic activity in vivo.
C26H33NO4 价格库存
MED14954 251565-85-2 Tesaglitazar
Tesaglitazar
双特异性PPARα/γ激动剂,Tesaglitazar 是一种过氧物酶体 PPAR alpha/gamma 受体的双重激动剂,对 PPARγ 的作用比 PPARα 强,对大鼠和人类 PPARα 作用的 EC50 分别为 13.4 μM 和 3.6 μM,对大鼠和人类 PPARγ 作用的 EC50 为 0.2 μM。
C20H24O7S 价格库存
MED14952 353280-43-0 S26948
S26948
PPARγ激动剂
C28H25NO7S 价格库存
MED14947 1014691-61-2 GSK 0660
GSK 0660
PPARδ拮抗剂,GSK0660是有效的 PPARβ 和 PPARδ 拮抗剂,IC50 均为159 nM。
C19H18N2O5S2 价格库存