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产品图片 产品编号 CAS号 产品名称 分子式 购物车
MED18542 66-71-7 o-Phenanthroline
o-Phenanthroline

o-Phenanthroline (1,10-Phenanthroline) 是一种金属螯合剂,可防止链脲佐菌素诱导染色体畸变。o-Phenanthroline (1,10-Phenanthroline)与Fe2+形成红色螯合物,在510 nm处最大吸收。

C12H8N2 价格库存
MED18525 947303-87-9 PF 429242
PF 429242
甾醇调节元件结合蛋白(SREBP)位点1蛋白酶抑制剂,PF-429242 is a potent inhibitor of S1P(cellular proprotein convertase sterol regulatory element-binding protein (SREBP) site 1 protease)
C25H35N3O2 价格库存
MED18536 185213-03-0 Butabindide oxalate
Butabindide oxalate
CCK失活丝氨酸蛋白酶(三肽基肽酶II)抑制剂,Butabindide is a potent inhibitor of cholecystokinin-inactivating peptidase/tripeptidyl peptidase 2 (CCK-inactivating peptidase/TPP-2; Ki = 7 nM).1 It is selective for CCK-inactivating peptidase/TPP-2 over a panel of serine proteases (Kis = >1 μM) as well as CCK receptors (Kis = >0.1 mM).
C17H25N3O2.C2H2O4 价格库存
MED18524 261619-50-5 CGS 35066
CGS 35066
内皮素转化酶(ECE)抑制剂
价格库存
MED18529 673202-67-0 Hexa-D-arginine
Hexa-D-arginine
弗林蛋白酶抑制剂,Hexa-D-arginine 是一种 furin 抑制剂。
C36H75N25O6 价格库存
MED18526 150113-99-8 Decanoyl-RVKR-CMK
Decanoyl-RVKR-CMK

枯草杆菌蛋白酶/Kex2p样前蛋白转化酶抑制剂,Furin inhibitor I is a selective, irreversible, and cell-permeable competitive inhibitor of proprotein convertases, including furin/SPC1 (Ki = ~1 nM), SPC2/PC2 (Ki = 0.36 nM), SPC3/PC1/PC3 (Ki = 2.0 nM), SPC4/PACE4 (Ki = 3.6 nM), SPC6/PC5/PC6, and SPC7/LP

C34H66CLN11O5 价格库存
MED18523 146794-84-5 Y-29794 oxalate
Y-29794 oxalate
价格库存
MED18530 697797-51-6 UAMC 00039 dihydrochloride
UAMC 00039 dihydrochloride
二肽基肽酶II(DPP-II)抑制剂,UAMC00039 dihydrochloride是高效,可逆,竞争性的dipeptidyl peptidase II抑制剂,IC50值为0.48 nM。
C16H26CL3N3O 价格库存
MED18527 1160928-63-1 RETF-4NA
RETF-4NA
糜酶底物肽,RETF-4NA 是糜蛋白酶的一个敏感的、特异性底物。
价格库存
MED18519 164204-38-0 Phosphoramidon (sodium salt)
Phosphoramidon (sodium salt)

Phosphoramidon (sodium salt) 是金属蛋白酶 ( metalloprotease ) 抑制剂 。抑制内皮素转化酶 ( ECE ) ,中性肽内切酶 ( NEP ) 和血管紧张素转换酶 ( ACE ) 的IC50 值分别为 3.5 ,0.034 和 78 μM。

C23H32N3NA2O10P 价格库存
MED18403 541503-81-5 Vicriviroc Malate
Vicriviroc Malate
第二代口服CCR5拮抗剂,Vicriviroc Malate is a potent, highly selective, and orally bioavailable CCR5 antagonist.
C28H38F3N5O2.C4H6O5 价格库存