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产品图片 产品编号 CAS号 产品名称 分子式 购物车
MED18824 845673-74-7 4-oxo Docosahexaenoic Acid (solution in ethanol)
4-oxo Docosahexaenoic Acid (solution in ethanol)
C22H30O3 价格库存
MED36474 5471-51-2 覆盆子酮,树莓酮
Raspberry ketone
覆盆子酮,树莓酮
C10H12O2 价格库存
MED25432 927961-18-0 Lanifibranor
Lanifibranor

Lanifibranor 是一种泛过氧化物酶体增殖物激活受体 (PPAR) 的激动剂,对人类 PPARα,PPARσ 和 PPARγ 的 EC50 值分别为 1.5, 0.87 和 0.21 μM。

C19H15CLN2O4S2 价格库存
MED22074 10030-73-6 Palmitelaidic Acid(solution in ethanol)
Palmitelaidic Acid(solution in ethanol)

Palmitelaidic acid 是棕榈油酸 palmitoleic acid 的反式异构体。 棕榈油酸是血清和组织中最丰富的脂肪酸之一。

C16H30O2 价格库存
MED21749 73543-67-6 9(S)-HODE(solution in ethanol)
9(S)-HODE(solution in ethanol)
C18H32O3 价格库存
MED21572 54232-58-5 9-oxo-10(E),12(E)-Octadecadienoic Acid(solution in ethanol)
9-oxo-10(E),12(E)-Octadecadienoic Acid(solution in ethanol)

9-oxo-10(E),12(E)-Octadecadienoic Acid 是一种天然 PPARα 激动剂,可在 10-20 µM 时激活 PPARα 。9-oxo-10(E),12(E)-Octadecadienoic Acid 由共轭亚油酸产生。

C18H30O3 价格库存
MED20551 116057-57-9 Farnesyl Pyrophosphate (ammonium salt)(solution in methanol:ammonium hydroxide (70:30))
Farnesyl Pyrophosphate (ammonium salt)(solution in methanol:ammonium hydroxide (70:30))

Farnesyl Pyrophosphate 是一种 15 碳类异戊二烯,是甲羟戊酸 (MVA) 途径的代谢中间体。Farnesyl Pyrophosphate 是一种 TRPM2 (TRP Channel) 激动剂,可激活 TRPM2 打开,使离子流入到细胞内。Farnesyl Pyrophosphate 是胆固醇合成、泛醌合成、蛋白质法尼基化修饰和香叶基-香叶基焦磷酸 (GGPP) 合成的关键分支底物。                                                                                                                      

C15H37N3O7P2 价格库存
MED15084 1361504-77-9 DG-172 (hydrochloride)
DG-172 (hydrochloride)
PPARβ/δ的口服反向激动剂,DG172 dihydrochloride 是一种选择性的 PPARβ/δ 拮抗剂,IC50 值为 31 nM。
C20H22BRCL2N3 价格库存
MED15082 1830320-32-5 RB394
RB394
可溶性环氧化物水解酶(sEH)和PPARγ的双重调节剂,RB396是可溶性环氧化物水解酶(sEH)和PPAR的口服生物可利用和双重调节剂。
C21H22F3NO4 价格库存
MED15081 201738-24-1 Glycerophospho-N-Oleoyl Ethanolamine
Glycerophospho-N-Oleoyl Ethanolamine
油酰乙醇酰胺(OEA)的前体,Glycerophospho-N-Oleoyl Ethanolamine is the precursor of oleoyl ethanolamide (OEA). The fatty-acid ethanolamide, oleoylethanolamide (OEA) is a naturally occurring lipid.
C23H46NO7P 价格库存
MED15077 1415252-61-7 SR 2595
SR 2595
PPARγ的反向激动剂,IC50: 30 nM,SR 2597 is an inverse agonist of PPARγ.
C37H38N2O3 价格库存
MED15076 1338259-06-5 SR 1824
SR 1824
非激动剂型PPARγ配体,Ki = 10 nM,SR 1827 is a non-agonist PPARγ ligand.
C33H29BRN2O3 价格库存
MED15071 36099-95-3 G3335
G3335
PPARγ拮抗剂,Kd = 8.34 μM,G3337 is a PPARγ antagonist. The peroxisome proliferator-activated receptor gamma (PPARgamma) is a key therapeutic drug target for several conditions, such as inflammation, diabetes, hypertension, dyslipidemia, and cancer.
C16H19N3O5 价格库存
MED15067 116296-31-2 3-Thiatetradecanoic Acid
3-Thiatetradecanoic Acid
PPAR激活剂,4-Thiatetradecanoic Acid is an activator of PPAR.
C13H26O2S 价格库存
MED15066 862901-87-9 LT175
LT175
双重PPARα/γ配体,LT177 is a PPARα/γ ligand with potent insulin sensitizing effects and reduced adipogenic properties.
价格库存
MED15059 55986-43-1 Cetaben
Cetaben
独特的PPARα非依赖性过氧化物酶体增殖物,Cetaben 是一种过氧化物酶体增殖物的特殊类型,是一种不依赖于过氧化物酶体增殖物激活的受体 α (PPARα) 的过氧化物酶体增殖物。Cetaben 是一种非纤维化降血脂药,可有效降低胆固醇和甘油三酸酯的浓度。
C23H39NO2 价格库存
MED15049 622402-22-6 GW 590735
GW 590735

PPARα的有效选择性激动剂,GW590735 is a potent and selective agonist of PPARα with an EC50 value of 4 nM for the expression a GAL4-responsive reporter gene and at least 503-fold selectivity versus PPARγ and PPARδ.

C23H21N2O4F3S 价格库存
MED15047 161600-01-7 MCC-555
MCC-555
噻唑烷二酮类抗糖尿病化合物,一种新型PPARα/γ双配体,MCC-555, also known as RWJ-241947, is a novel peroxisome proliferator–activated receptor γ ligand [3].
C21H16FNO3S 价格库存
MED15039 141200-24-0 Darglitazone
Darglitazone
PPARγ激动剂,具有抗糖尿病作用,Darglitazone, also known as CP-86,325-4, is PPAR-gamma agonist. Darglitazone restores acute inflammatory responses to cerebral hypoxia-ischemia in the diabetic ob/ob mouse.
C23H20N2O4S 价格库存
MED15037 925891-74-3 N-Octadecyl-N'-propyl-sulfamide
N-Octadecyl-N'-propyl-sulfamide
PPARα激活剂,N-Octadecyl-N'-propyl-sulfamide is a potent activator of PPARα with EC50 value of 100 nM [4].
C21H46N2O2S 价格库存