1-Palmitoyl-2-linoleoyl PE (PLPE) is one of the many phosphatidylethanolamines that may be present in cellular membranes. It has been used in studies involving the biosynthesis of anandamide via the phospholipase A₂ (PLA₂) and lysoPLD pathways. PLPE can also be used as a specific substrate to assess the activity of sPLA₂-IIA in the presence of other phospholipids.

ONO-RS-082是Ca2+-依赖性磷脂酶A2的可逆抑制剂

磷脂酶D（PLD）抑制剂，Halopemide 是一种有效的磷脂酶 D (PLD) 抑制剂，对人 PLD1 和 PLD2 的 IC50 分别为 220 和 312 nM。Halopemide 是多巴胺受体拮抗剂，是一种精神药物。

分泌型磷脂酶A2（sPLA2）抑制剂，LY 311727 is a specific group II sPLA2 (phospholipase A2 (PLA3)) inhibitor which has been reported to attenuate VEGF-mediated platelet-activating factor (PAF) synthesis in HUVEC and BAEC cells.

抑制磷脂酰肌醇磷脂酶C，Edelfosine is a synthetic lysophospholipid analog that selectively inhibits PLC with IC50 of 9.8 uM in fibroblasts and adenocarcinoma cells.