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产品图片 产品编号 CAS号 产品名称 分子式 购物车
MED11838 2491-38-5 PTP Inhibitor I
PTP Inhibitor I
酪氨酸磷酸酶(PTP)抑制剂,4'-bromo-Resveratrol is a Sirt1 and Sirt3 inhibitor.Sirtuins are protein deacetylases regulating aging processes and many physiological functions. Resveratrol activates human Sirt1 and inhibits Sirt3, and can mimic calorie restriction effects including lifespan extension in lower organisms.
C8H7BRO2 价格库存
MED11727 78111-17-8 Okadaic acid(solution)
Okadaic acid(solution)
Okadaic acid 是从 Halichondria 属的黑色海绵中提取的。Okadaic acid 是一种非竞争性,选择性和可逆的丝氨酸/苏氨酸特异性蛋白磷酸酶 1 (PP1),PP2A 和 PP3 的抑制剂,IC50 分别为 10-15 nM,0.5 nM 和 4 nM。Okadaic acid 通过细胞凋亡消除后生共生体/寄生虫
C44H68O13 价格库存
MED11726 249537-73-3 NFAT Inhibitor
NFAT Inhibitor
NFAT Inhibitor 是一种选择性的 NFAT 抑制剂。Selective inhibitor of calcineurin-mediated dephosphorylation of nuclear factor of activated T cells (NFAT). Does not disrupt other calcineurin-dependent pathways. Inhibits NFAT activation and NFAT-dependent expression of endogenous cytokine genes in T cells.
C75H118N20O22S 价格库存
MED11846 893449-38-2 PRL-3 Inhibitor
PRL-3 Inhibitor

再生肝脏蛋白磷酸酶-3(PRL-3)抑制剂,BR-1 is a PRL-3 inhibitor which blocks the migration and invasion of metastatic cancer cells.

C17H11BR2NO2S2 价格库存
MED11854 329317-98-8 PTP Inhibitor IV
PTP Inhibitor IV
PTP抑制剂,IC50: 1.8, 2.5, 8.4, 13, 20, 6.4, and 6.7 μM for SHP-2, PTP1B, PTP-ε, PTP-Meg-2, PTP-σ, PTP-β, and PTP-μ, respectively PTP Inhibitor IV is a protein tyrosine phosphatases (PTPs) inhibitor.
价格库存
MED11856 722494-26-0 bpV(HOpic) (potassium salt, technical grade)
bpV(HOpic) (potassium salt, technical grade)
蛋白酪氨酸磷酸酶(PTPs)抑制剂,BpV(HOpic) 是一种有效的和选择性的 PTEN 抑制剂,IC50 值为 14 nM。Nanocarrier-BpV(HOpic) 具有神经保护作用。
价格库存
MED11853 13408-09-8 β-Glycerophosphate (sodium salt hydrate)
β-Glycerophosphate (sodium salt hydrate)
蛋白磷酸酶抑制剂,β-Glycerol phosphate disodium salt pentahydrate 是磷酸酶和张力蛋白同源物 (PTEN) 的抑制剂,来自专利US 20110002877 A1。
C3H7NA2O6P 价格库存
MED11845 1465-77-6 Cantharidic Acid (sodium salt)
Cantharidic Acid (sodium salt)
PP1和PP2A抑制剂,Cantharidic acid, an inhibitor of protein phosphatases, is first isolated from Chinese blister beetles. Cantharidic acid is a hydrolysis product of cantharidin.
C10H12O5-2.2[NA+] 价格库存
MED11812 383907-43-5 NSC 663284
NSC 663284
Cdc25双特异性磷酸酶抑制剂,NSC 663284是 Cdc25 双重特异性磷酸酶抑制剂, IC50 值为0.21 μM
C15H16CLN3O3 价格库存
MED11837 2632-13-5 PTP Inhibitor II
PTP Inhibitor II
蛋白酪氨酸磷酸酶(PTP)抑制剂,PTP inhibitor 1 是一种蛋白酪氨酸磷酸酶 (PTP) 抑制剂,具有抗血管生成活性。
C9H9BRO2 价格库存
MED11811 93718-83-3 NSC 95397
NSC 95397
NSC 95397 是一种双特异性磷酸酶抑制剂,抑制丝裂原活化蛋白激酶磷酸酶-1 (MKP-1)。NSC 95397 通过 MKP-1 和 ERK1/2 途径抑制结肠癌细胞的增殖并诱导细胞凋亡。
C14H14O4S2 价格库存
MED11814 119757-73-2 Tautomycetin
Tautomycetin
蛋白磷酸酶(PP)1抑制剂
C33H50O10 价格库存
MED11789 5578-73-4 Sanguinarine chloride
Sanguinarine chloride
PP2C和MKP-1抑制剂,Sanguinarine chloride是一种强效的和特异性的PP2C抑制剂,Ki值为0.68 μM,也是一种选择性的具细胞活性的MKP-1抑制剂,IC50值为10 μM.Sanguinarine也是一种AMPK变构激活剂
C20H14CLNO4 价格库存
MED11737 638156-11-3 CID 2011756
CID 2011756
CID-2011756是蛋白激酶D1(PKD1)的新型强效抑制剂,PKD1是丝氨酸/苏氨酸激酶新家族的3种PKD亚型之一,参与细胞增殖、存活、侵袭和蛋白转运,体外IC50值为3.2 μM。CID-2011756可以抑制pan-PKD的活性,与ATP竞争抑制PKD2和PDK3,IC50分别为0.6 μM和0.7 μM。研究结果表明,CID-2011756是一种具细胞活性的PKD1抑制剂,在LNCaP前列腺癌细胞中,以浓度依赖性方式抑制佛波酯诱导的内源性PKD1活化,EC50值为10 μM
C22H21N2O3CL 价格库存
MED11741 13098-73-2 Sephin1
Sephin1
Sephin1 is a selective inhibitor of stress-induced PPP1R15A and targets disease associated with accumulation of misfolded protein
C8H9N4CL 价格库存
MED11749 81525-10-2 Nafamostat
Nafamostat

Nafamostat是广谱的丝氨酸蛋白酶抑制剂,血管舒缓素抑制剂,能抑制血液凝固,还是潜在的补体抑制剂。Nafamostat, a synthetic serine protease inhibitor, is an anticoagulant.

C19H17N5O2 价格库存
MED11722 20263-06-3 DL-AP3
DL-AP3
谷氨酸受体拮抗剂和HPSP抑制剂,Competitive group I metabotropic glutamate receptor antagonist and inhibitor of phosphoserine phosphatase.
C3H8NO5P 价格库存
MED11720 101932-71-2 Calyculin A
Calyculin A
CaMKII抑制剂,Calcineurin autoinhibitory peptide 是一种选择性的 Ca2+/ 钙调蛋白依赖性蛋白磷酸酶(钙调神经磷酸酶)的抑制剂,IC50 值大约为 10 μM。Calcineurin autoinhibitory peptide 可以保护神经元免受兴奋性神经元死亡
C50H81N4O15P 价格库存
MED11725 3519-82-2 INCA-6
INCA-6
Calcineurin-NFAT信号通路抑制剂,INCA-6是转录因子NFAT的选择性抑制剂,体外Kd值为0.8 mM[1]
C20H12O2 价格库存
MED11750 80251-32-7 Nafamostat hydrochloride
Nafamostat hydrochloride
合成的丝氨酸蛋白酶抑制剂,Nafamostat盐酸盐是广谱的丝氨酸蛋白酶抑制剂,血管舒缓素抑制剂,能抑制血液凝固,还是潜在的补体抑制剂。
C19H19CL2N5O2 价格库存