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产品图片 产品编号 CAS号 产品名称 分子式 购物车
MED19475 608512-97-6 西维因,PKR Inhibitor
PKR Inhibitor

双链RNA激活蛋白激酶(PKR)抑制剂,PKR-IN-C16 是特异性蛋白激酶 (PKR) 抑制剂。PKR-IN-C16 能够抑制 PKR 的自磷酸化,PKR 在原代神经元细胞培养中诱导的翻译阻断可被 PKR-IN-C16 解除。

C13H8N4OS 价格库存
MED19473 208445-06-1 Rp-8-bromo-Cyclic GMPS (sodium salt)
Rp-8-bromo-Cyclic GMPS (sodium salt)
cGMP依赖性蛋白激酶(cGK)抑制剂,Rp-8-bromo-Cyclic GMPS is a cGMP-dependent protein kinase (cGK) inhibitor.
价格库存
MED19474 208445-07-2 Rp-8-pCPT-Cyclic GMPS (sodium salt)
Rp-8-pCPT-Cyclic GMPS (sodium salt)

Rp-8-pCPT-Cyclic GMPS is a stable, cell-permeable cGMP analog that competitively inhibits cGMP-dependent protein kinases (cGKs), including cGK Iα and cGK II (IC50s = 18.3 and 0.16 µM, respectively). The pCPT (p-chlorophenylthio) group at the 8-position of the purine increases both enzyme affinity and membrane permeability over related compounds. At 10 µM, it blocks the relaxation of rat tail arteries induced by the nitric oxide donor SIN-1.

C16H14CLN5O6PS2.NA 价格库存
MED19484 210297-47-5 HA-100 (hydrochloride)
HA-100 (hydrochloride)
蛋白激酶(PKs)抑制剂,HA-100 is a dechlorinated analogue of 1-(8-chloro-5-isoquinolinesulfonyl)piperazine (HA-156). HA-100 is an inhibitor of protein kinases (PKs) including PKA, PKC, and PKG [1].
价格库存
MED19434 81156-93-6 RR-src
RR-src
酪氨酸激酶底物肽
C64H106N22O21 价格库存
MED19439 99533-80-9 K 252a
K 252a
蛋白激酶抑制剂,K-252a 可从土壤真菌Nocardiopsis sp.中分离得到的一种十字孢碱的类似物,是蛋白激酶的抑制剂,对 PKC、PKA、II型钙调素依赖性激酶和磷酸化酶激酶的 IC50 值分别为470 nM、140 nM、270 nM和1.7 nM。
C27H21N3O5 价格库存
MED19428 108930-17-2 H-7 dihydrochloride
H-7 dihydrochloride
蛋白激酶抑制剂,H7 is a specific protein kinase C inhibitor and protein kinase G inhibitor, which inhibits superoxide release from human neutrophils (PMN) stimulated with phorbol myristate acetate or synthetic diacylglycerol.
C14H19CL2N3O2S 价格库存
MED19398 116700-36-8 H-9 dihydrochloride
H-9 dihydrochloride
蛋白激酶抑制剂
C11H13N3O2S.2[HCL] 价格库存
MED19354 62996-74-1 Staurosporine
Staurosporine
蛋白激酶抑制剂,Staurosporine是一种有效,非选择性蛋白激酶抑制剂,抑制 PKC,PKA,c-Fgr,和 Phosphorylase kinase 的 IC50 分别为 6 nM,15 nM,2 nM,6 nM。
C28H26N4O3 价格库存