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产品图片 产品编号 CAS号 产品名称 分子式 购物车
MED16986 106469-57-2 Cyanopindolol hemifumarate
Cyanopindolol hemifumarate

Cyanopindolol hemifumarate 是5-HT1A/1B拮抗剂,也是一种 β-肾上腺素 受体拮抗剂。

C36H46N6O8 价格库存
MED17002 78095-19-9 (R)-(+)-8-Hydroxy-DPAT hydrobromide
(R)-(+)-8-Hydroxy-DPAT hydrobromide
5-HT1A 5-羟色胺受体激动剂
C16H26BRNO 价格库存
MED16980 159187-70-9 MM 77 dihydrochloride
MM 77 dihydrochloride
5-HT1A受体拮抗剂
价格库存
MED16973 157798-13-5 5-Nonyloxytryptamine oxalate
5-Nonyloxytryptamine oxalate

5-Nonyloxytryptamine oxalate 是一种有效的选择性 5-HT1B 受体激动剂。

C19H30N2O.C2H2O4 价格库存
MED16964 159651-91-9 8-Hydroxy-PIPAT oxalate
8-Hydroxy-PIPAT oxalate
5-HT1A受体激动剂
C16H22NOI.C4H4O4 价格库存
MED16955 99201-87-3 Anpirtoline hydrochloride
Anpirtoline hydrochloride
5-HT1B受体激动剂,Anpirtoline HCl is highly potent 5-HT1B receptor agonist which decreases central serotonin synthesis and attenuates aggressive behavior in vivo. Anpirtoline HCl also acts as an antagonist at 5-HT3 receptors and is brain penetrant. Anpirtoline is a receptor agonist with antinociceptive/antidepressant-like actions in rodents.
C10H13N2SCL.HCL 价格库存
MED16937 76135-31-4 8-Hydroxy-DPAT hydrobromide
8-Hydroxy-DPAT hydrobromide
5-HT1A激动剂,8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) 是一种有效的,选择性 5-HT1A 激动剂,pIC50 为 8.19。8-Hydroxy-DPAT hydrobromide 对 5-HT1 结合位点的亚型具有近 1000 倍的选择性。
C16H26BRNO 价格库存
MED16940 82900-57-0 BP 554 maleate
BP 554 maleate
5-HT1A激动剂
C20H24N2O3 价格库存
MED16945 109028-10-6 CGS 12066B dimaleate
CGS 12066B dimaleate
5-HT1B完全激动剂
C17H17N4F3.2[C4H4O4] 价格库存
MED16939 115338-32-4 NAN-190 hydrobromide
NAN-190 hydrobromide

5-HT1A拮抗剂,NAN-190溴酸盐是一种血清素受体5-HT受体拮抗剂, NAN-190是5-HT 1A选择性拮抗剂。

C23H28BRN3O3 价格库存
MED16927 102908-60-1 MDL 73005EF hydrochloride
MDL 73005EF hydrochloride
5-HT1A受体拮抗剂
价格库存
MED16928 113777-40-5 MDL 72832 hydrochloride
MDL 72832 hydrochloride
5-HT1A受体的配体
价格库存
MED16855 448904-47-0 WY 45233 succinate
WY 45233 succinate
5-羟色胺和去甲肾上腺素再摄取抑制剂
C16H25NO2.C4H6O4 价格库存
MED16846 184674-99-5 NAD 299 hydrochloride
NAD 299 hydrochloride

NAD-299 HCl 是高亲和力5-HT1A受体拮抗剂。

C18H23FN2O2.HCL 价格库存
MED16817 103628-46-2 Sumatriptan
Sumatriptan
5-HT1受体激动剂,用作偏头痛治疗药,为5-羟色胺受体活动药,主要作用方式为选择性地收缩颅侧血管。用于偏头痛。
C14H21N3O2S 价格库存
MED16833 84484-78-6 BTS 54-505 hydrochloride
BTS 54-505 hydrochloride
C15H23CL2N 价格库存
MED16783 607742-69-8 SB742457
SB742457
5-HT6受体拮抗剂,具有高选择性和高亲和力。SB742457是5-HT6受体拮抗剂,pKi为9.63,比对其它受体的抑制性高100倍以上。
C19H19N3O2S 价格库存
MED16773 64887-14-5 Urapidil HCl
Urapidil HCl
α1肾上腺素受体拮抗剂和5-HT1A受体激动剂,Urapidil盐酸盐是α1-肾上腺素受体拮抗剂和5-HT1A受体激动剂。
C20H30CLN5O3 价格库存
MED16765 123040-16-4 Azasetron HCl
Azasetron HCl
5-HT3受体拮抗剂,Azasetron盐酸盐是5-HT3受体选择性拮抗剂,IC50为0.33 nM。
C17H21CL2N3O3 价格库存
MED16755 5053-08-7 Fenspiride HCl
Fenspiride HCl
α肾上腺素能和H1组胺受体拮抗剂,Fenspiride盐酸盐是肾上腺素能受体和H1受体拮抗剂。
C15H21CLN2O2 价格库存