LY 456236 hydrochloride

LY 456236 hydrochloride (订货以CAS编码或英文名称为准)

mGlu1受体拮抗剂,LY456236 HCl is a selective mGlu1 receptor antagonist (IC50 values are 143 nM and > 10 μM for mGlu1 and mGlu5 receptors respectively).
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编号:MED17076
分子式:C16H16CLN3O2
CAS号:338736-46-2
分子量:317.77
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英文名称: LY 456236 hydrochloride
英文别名: LY 456236;6-Methoxy-N-(4-methoxyphenyl)-4-quinazolinamine hydrochloride (1: 1);LY 456236 hydrochloride;(4-Methoxy-phenyl)-(6-methoxy-quinazolin-4-yl)-amine hydrochloride;6-Methoxy-N-(4-methoxyphenyl)-4-quinazolinamine hydrochloride;LY456236;MPMQ
CAS号: 338736-46-2
分子式: C16H16CLN3O2
分子量: 317.77
mGlu1受体拮抗剂,LY456236 HCl is a selective mGlu1 receptor antagonist (IC50 values are 143 nM and > 10 μM for mGlu1 and mGlu5 receptors respectively). LY456236 HCl reduces hyperalgesic behavior induced by formalin in both mouse and rat with ED50 values of 28 and 16.3 mg/kg respectively. 产品性质
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